Vol. 9 No. 4 (2021) | ADMET and DMPK

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href="https://pub.iapchem.org/ojs/index.php/admet/login"> Login </a> </li> </ul> </div> </nav> </div> </header> <div class="pkp_structure_content has_sidebar"> <div class="pkp_structure_main" role="main"> <a id="pkp_content_main"></a> <div class="page page_issue"> <nav class="cmp_breadcrumbs" role="navigation" aria-label="You are here:"> <ol> <li> <a href="https://pub.iapchem.org/ojs/index.php/admet/index"> Home </a> <span class="separator">/</span> </li> <li> <a href="https://pub.iapchem.org/ojs/index.php/admet/issue/archive"> Archives </a> <span class="separator">/</span> </li> <li class="current" aria-current="page"> <span aria-current="page"> Vol. 9 No. 4 (2021) </span> </li> </ol> </nav> <div class="current_issue_title admet_toc_issue_title"> Vol. 9 No. 4 (2021) </div> <div class="obj_issue_toc"> <div class="heading"> <div class="description"> <p><strong>New Therapeutic Modalities in Drug Discovery and Development: Insights & Opportunities </strong></p> <p><strong>Special issue</strong> guest-edited by <em>Manfred Kansy</em> and <em>Giulia Caron</em></p> </div> <div class="published"> <span class="label"> Published: </span> <span class="value"> 15-12-2021 </span> </div> </div> <div class="sections"> <div class="section"> <h2> Editorial </h2> <ul class="cmp_article_list articles"> <li> <div class="obj_article_summary"> <div class="admet_article_summ"> <h3 class="title"> <a id="article-1209" href="https://pub.iapchem.org/ojs/index.php/admet/article/view/1209"> New therapeutic modalities in drug discovery and development: Insights & opportunities </a> </h3> <div class="meta"> <div class="authors"> Manfred Kansy, Giulia Caron </div> <div class="admet_meta_pages"> ADMET and DMPK, Vol. 9 No. 4 (2021), 227-230 </div> <div class="published"> <div class="admet_published">Published 15-12-2021;</div> <div class="admet_doi item doi"> <span class="label"> DOI: </span> <span class="value"> <a href="https://doi.org/10.5599/admet.1209"> https://doi.org/10.5599/admet.1209 </a> </span> </div> </div> </div> <ul class="galleys_links"> <li> <a class="obj_galley_link pdf" href="https://pub.iapchem.org/ojs/index.php/admet/article/view/1209/1379" aria-labelledby=article-1209> PDF </a> </li> </ul> </div> <div class="cover toc_cover_admet"> <a href="https://pub.iapchem.org/ojs/index.php/admet/article/view/1209" class="file"> <img src="https://pub.iapchem.org/ojs/public/journals/4/article_1209_cover_en_US.png" alt="New therapeutic modalities"> </a> </div> </div> <hr class="toc_hr_admet" /> </li> </ul> </div> <div class="section"> <h2> Reviews </h2> <ul class="cmp_article_list articles"> <li> <div class="obj_article_summary"> <div class="admet_article_summ"> <h3 class="title"> <a id="article-951" href="https://pub.iapchem.org/ojs/index.php/admet/article/view/951"> Current state and future of 3D bioprinted models for cardio-vascular research and drug development </a> </h3> <div class="meta"> <div class="authors"> Liudmila Polonchuk, Carmine Gentile </div> <div class="admet_meta_pages"> ADMET and DMPK, Vol. 9 No. 4 (2021), 231-242 </div> <div class="published"> <div class="admet_published">Published 25-08-2021;</div> <div class="admet_doi item doi"> <span class="label"> DOI: </span> <span class="value"> <a href="https://doi.org/10.5599/admet.951"> https://doi.org/10.5599/admet.951 </a> </span> </div> </div> </div> <ul class="galleys_links"> <li> <a class="obj_galley_link pdf" href="https://pub.iapchem.org/ojs/index.php/admet/article/view/951/1315" aria-labelledby=article-951> PDF </a> </li> </ul> </div> <div class="cover toc_cover_admet"> <a href="https://pub.iapchem.org/ojs/index.php/admet/article/view/951" class="file"> <img src="https://pub.iapchem.org/ojs/public/journals/4/article_951_cover_en_US.jpg" alt="3D bioprinted models for cardio-vascular research and drug development"> </a> </div> </div> <hr class="toc_hr_admet" /> </li> </ul> </div> <div class="section"> <h2> Original Scientific Articles </h2> <ul class="cmp_article_list articles"> <li> <div class="obj_article_summary"> <div class="admet_article_summ"> <h3 class="title"> <a id="article-1037" href="https://pub.iapchem.org/ojs/index.php/admet/article/view/1037"> Are we ready to design oral PROTACs®? </a> </h3> <div class="meta"> <div class="authors"> Diego Garcia Jimenez, Matteo Rossi Sebastiano, Giulia Caron, Giuseppe Ermondi </div> <div class="admet_meta_pages"> ADMET and DMPK, Vol. 9 No. 4 (2021), 243-254 </div> <div class="published"> <div class="admet_published">Published 31-08-2021;</div> <div class="admet_doi item doi"> <span class="label"> DOI: </span> <span class="value"> <a href="https://doi.org/10.5599/admet.1037"> https://doi.org/10.5599/admet.1037 </a> </span> </div> </div> </div> <ul class="galleys_links"> <li> <a class="obj_galley_link pdf" href="https://pub.iapchem.org/ojs/index.php/admet/article/view/1037/1316" aria-labelledby=article-1037> PDF </a> </li> <li> <a class="obj_galley_link pdf" href="https://pub.iapchem.org/ojs/index.php/admet/article/view/1037/1317" aria-labelledby=article-1037> Supplementary material </a> </li> </ul> </div> <div class="cover toc_cover_admet"> <a href="https://pub.iapchem.org/ojs/index.php/admet/article/view/1037" class="file"> <img src="https://pub.iapchem.org/ojs/public/journals/4/article_1037_cover_en_US.jpg" alt="Oral PROTAC"> </a> </div> </div> <hr class="toc_hr_admet" /> </li> <li> <div class="obj_article_summary"> <div class="admet_article_summ"> <h3 class="title"> <a id="article-1023" href="https://pub.iapchem.org/ojs/index.php/admet/article/view/1023"> Synthesis of silymarin−selenium nanoparticle conjugate and examination of its biological activity in vitro </a> </h3> <div class="meta"> <div class="authors"> Sergey Staroverov, Sergey Kozlov, Alexander Fomin, Konstantin Gabalov, Vitaliy Khanadeev, Dmitry Soldatov, Ivan Domnitsky, Lev Dykman, Sergey V. Akchurin, Olga Guliy </div> <div class="admet_meta_pages"> ADMET and DMPK, Vol. 9 No. 4 (2021), 255-266 </div> <div class="published"> <div class="admet_published">Published 14-11-2021;</div> <div class="admet_doi item doi"> <span class="label"> DOI: </span> <span class="value"> <a href="https://doi.org/10.5599/admet.1023"> https://doi.org/10.5599/admet.1023 </a> </span> </div> </div> </div> <ul class="galleys_links"> <li> <a class="obj_galley_link pdf" href="https://pub.iapchem.org/ojs/index.php/admet/article/view/1023/1341" aria-labelledby=article-1023> PDF </a> </li> </ul> </div> <div class="cover toc_cover_admet"> <a href="https://pub.iapchem.org/ojs/index.php/admet/article/view/1023" class="file"> <img src="https://pub.iapchem.org/ojs/public/journals/4/article_1023_cover_en_US.jpg" alt="Silymarin-selenium nanoparticle conjugates"> </a> </div> </div> <hr class="toc_hr_admet" /> </li> <li> <div class="obj_article_summary"> <div class="admet_article_summ"> <h3 class="title"> <a id="article-1034" href="https://pub.iapchem.org/ojs/index.php/admet/article/view/1034"> cΔlog kwIAM: can we afford estimation of small molecules’ blood-brain barrier passage based upon in silico phospholipophilicity? </a> </h3> <div class="meta"> <div class="authors"> Lucia Grumetto, Giacomo Russo </div> <div class="admet_meta_pages"> ADMET and DMPK, Vol. 9 No. 4 (2021), 267-281 </div> <div class="published"> <div class="admet_published">Published 15-12-2021;</div> <div class="admet_doi item doi"> <span class="label"> DOI: </span> <span class="value"> <a href="https://doi.org/10.5599/admet.1034"> https://doi.org/10.5599/admet.1034 </a> </span> </div> </div> </div> <ul class="galleys_links"> <li> <a class="obj_galley_link pdf" href="https://pub.iapchem.org/ojs/index.php/admet/article/view/1034/1370" aria-labelledby=article-1034> PDF </a> </li> <li> <a class="obj_galley_link pdf" href="https://pub.iapchem.org/ojs/index.php/admet/article/view/1034/1380" aria-labelledby=article-1034> Supplementary data </a> </li> </ul> </div> <div class="cover toc_cover_admet"> <a href="https://pub.iapchem.org/ojs/index.php/admet/article/view/1034" class="file"> <img src="https://pub.iapchem.org/ojs/public/journals/4/article_1034_cover_en_US.jpg" alt="Blood-Brain Barrier passage of small molecules"> </a> </div> </div> <hr class="toc_hr_admet" /> </li> </ul> </div> </div> </div> </div> </div> <div class="pkp_structure_sidebar left" role="complementary" aria-label="Sidebar"> <div class="pkp_block block_custom" id="customblock-jif"> <h2 class="title pkp_screen_reader">JIF</h2> <div class="content"> <p><img src="https://pub.iapchem.org/ojs/public/site/images/editorial/clarivate-analytics-logo.svg-d36ab472132a0b58eedd4e6a6746fc3c.png" alt="" width="175" height="31"><br><img src="https://pub.iapchem.org/ojs/public/site/images/editorial/snimak-ekrana-2024-06-21-102313.png" alt="" width="215" height="73"></p> <p><img src="https://pub.iapchem.org/ojs/public/site/images/editorial/mceclip0-639ce01c3d3bc312dbd548e85e2889bf.png" width="390" height="128"><br><img src="https://pub.iapchem.org/ojs/public/site/images/editorial/mceclip1-aaf59f2587d45bc7e184c2349f65948b.png" width="400" height="129"></p> </div> </div> <div class="pkp_block block_custom" id="customblock-elsevier"> <h2 class="title pkp_screen_reader">elsevier</h2> <div class="content"> <div style="height: 100px; 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Vol. 9 No. 4 (2021) | ADMET and DMPK