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Search results for: N-[3-(2-Benzothiazolyl)-4-methylthiazol-2(3H)-ylidene]benzamides
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class="card-body"><strong>Edition:</strong> International</div> </div> </div> <div class="col-sm-3"> <div class="card"> <div class="card-body"><strong>Paper Count:</strong> 2</div> </div> </div> </div> <h1 class="mt-3 mb-3 text-center" style="font-size:1.6rem;">Search results for: N-[3-(2-Benzothiazolyl)-4-methylthiazol-2(3H)-ylidene]benzamides</h1> <div class="card paper-listing mb-3 mt-3"> <h5 class="card-header" style="font-size:.9rem"><span class="badge badge-info">2</span> Design and Synthesis of Novel Benzamides as Non-Ulcerogenic Anti-Inflammatory Agents</h5> <div class="card-body"> <p class="card-text"><strong>Authors:</strong> <a href="https://publications.waset.org/abstracts/search?q=Khadse%20Saurabh">Khadse Saurabh</a>, <a href="https://publications.waset.org/abstracts/search?q=Talele%20Gokul"> Talele Gokul</a>, <a href="https://publications.waset.org/abstracts/search?q=Surana%20Sanjay"> Surana Sanjay</a> </p> <p class="card-text"><strong>Abstract:</strong></p> In an endeavor to find a new class of anti-inflammatory agents, a series of novel benzamides (ab1-ab16) were synthesized by utilizing some arylideneoxazolones (az1-az4) having 2-acetyloxyphenyl substitution on their second position. Structures of these synthesized compounds were confirmed by IR, 1H-NMR, 13C NMR, and HRMS. Among the tested benzamide compounds 3ab1, 3ab2, 3ab11, and 3ab16 showed promising anti-inflammatory activity with lessened propensity to cause gastro-intestinal hypermotility and ulceration when compared with standard Indomethacin. Virtual screening was performed by docking the designed compounds into the ATP binding site of COX-2 receptor to predict if these compounds have analogous binding mode to the COX-2 inhibitor. <p class="card-text"><strong>Keywords:</strong> <a href="https://publications.waset.org/abstracts/search?q=benzamides" title="benzamides">benzamides</a>, <a href="https://publications.waset.org/abstracts/search?q=anti-inflammatory" title=" anti-inflammatory"> anti-inflammatory</a>, <a href="https://publications.waset.org/abstracts/search?q=gastro-intestinal%20hypermotility" title=" gastro-intestinal hypermotility"> gastro-intestinal hypermotility</a>, <a href="https://publications.waset.org/abstracts/search?q=ulcerogenic%20activity" title=" ulcerogenic activity"> ulcerogenic activity</a>, <a href="https://publications.waset.org/abstracts/search?q=docking" title=" docking "> docking </a> </p> <a href="https://publications.waset.org/abstracts/19186/design-and-synthesis-of-novel-benzamides-as-non-ulcerogenic-anti-inflammatory-agents" class="btn btn-primary btn-sm">Procedia</a> <a href="https://publications.waset.org/abstracts/19186.pdf" target="_blank" class="btn btn-primary btn-sm">PDF</a> <span class="bg-info text-light px-1 py-1 float-right rounded"> Downloads <span class="badge badge-light">440</span> </span> </div> </div> <div class="card paper-listing mb-3 mt-3"> <h5 class="card-header" style="font-size:.9rem"><span class="badge badge-info">1</span> Efficient Synthesis of Benzothiazolyl Thioureas Based Thiazoline Heterocycles</h5> <div class="card-body"> <p class="card-text"><strong>Authors:</strong> <a href="https://publications.waset.org/abstracts/search?q=Hummera%20Rafique">Hummera Rafique</a>, <a href="https://publications.waset.org/abstracts/search?q=Aamer%20Saeed"> Aamer Saeed</a> </p> <p class="card-text"><strong>Abstract:</strong></p> 2-Aminobenzothiazoles are highly biologically active compounds, as many important applications are associated with this nucleus. They serve as precursors for the synthesis of thioureas. Benzothiazolyl thioureas are exceptionally versatile building blocks towards the synthesis of a wide variety of heterocyclic systems, which also possess extensive range of bioactivities. These thioureas were converted into five-membered heterocycles with imino moiety like N-[3-(2-Benzothiazolyl)-4-methylthiazol-2(3H)-ylidene] benzamides by base-catalyzed cyclization of corresponding thioureas with 2-bromoacetone and triethylamine in good yields. <p class="card-text"><strong>Keywords:</strong> <a href="https://publications.waset.org/abstracts/search?q=N-%5B3-%282-Benzothiazolyl%29-4-methylthiazol-2%283H%29-ylidene%5Dbenzamides" title="N-[3-(2-Benzothiazolyl)-4-methylthiazol-2(3H)-ylidene]benzamides">N-[3-(2-Benzothiazolyl)-4-methylthiazol-2(3H)-ylidene]benzamides</a>, <a href="https://publications.waset.org/abstracts/search?q=1-%28substitutedbenzo%5Bd%5D%20thiazol-2-yl%29-3-aroylthioureas" title=" 1-(substitutedbenzo[d] thiazol-2-yl)-3-aroylthioureas"> 1-(substitutedbenzo[d] thiazol-2-yl)-3-aroylthioureas</a>, <a href="https://publications.waset.org/abstracts/search?q=2-aminobenzothiazoles" title=" 2-aminobenzothiazoles"> 2-aminobenzothiazoles</a>, <a href="https://publications.waset.org/abstracts/search?q=antibacterial%20activities" title=" antibacterial activities"> antibacterial activities</a> </p> <a href="https://publications.waset.org/abstracts/22525/efficient-synthesis-of-benzothiazolyl-thioureas-based-thiazoline-heterocycles" class="btn btn-primary btn-sm">Procedia</a> <a href="https://publications.waset.org/abstracts/22525.pdf" target="_blank" class="btn btn-primary btn-sm">PDF</a> <span class="bg-info text-light px-1 py-1 float-right rounded"> Downloads <span class="badge badge-light">340</span> </span> </div> </div> </div> </main> <footer> <div id="infolinks" class="pt-3 pb-2"> <div class="container"> <div style="background-color:#f5f5f5;" class="p-3"> <div class="row"> <div class="col-md-2"> <ul class="list-unstyled"> About <li><a href="https://waset.org/page/support">About Us</a></li> <li><a href="https://waset.org/page/support#legal-information">Legal</a></li> <li><a target="_blank" rel="nofollow" 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